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A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer
Fabrizio Pertusati,
Salvatore Ferla
,
Marcella Bassetto,
Andrea Brancale,
Sahar Khandil,
Andrew D. Westwell,
Christopher McGuigan
European Journal of Medicinal Chemistry, Volume: 180, Pages: 1 - 14
Swansea University Authors:
Salvatore Ferla , Marcella Bassetto
Full text not available from this repository: check for access using links below.
DOI (Published version): 10.1016/j.ejmech.2019.07.001
Abstract
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer
Published in: | European Journal of Medicinal Chemistry |
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ISSN: | 0223-5234 |
Published: |
Elsevier BV
2019
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URI: | https://cronfa.swan.ac.uk/Record/cronfa52218 |
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2019-10-01T20:18:38Z |
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2020-11-06T04:12:41Z |
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2020-11-05T17:09:52.0164718 v2 52218 2019-10-01 A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer d4c62248f510e3b221916989a7bbe6a6 0000-0002-5918-9237 Salvatore Ferla Salvatore Ferla true false b97beeed16f8e0524551233ade909565 Marcella Bassetto Marcella Bassetto true false 2019-10-01 PHAR Journal Article European Journal of Medicinal Chemistry 180 1 14 Elsevier BV 0223-5234 Pentafluorosulfanyl; Pentafluoroethyl; Prostate cancer; Androgen receptor; Antiproliferative activity; Enobosarm; Bicalutamide; Enzalutamide 15 10 2019 2019-10-15 10.1016/j.ejmech.2019.07.001 http://orca.cf.ac.uk/124785/ COLLEGE NANME Pharmacy COLLEGE CODE PHAR Swansea University 2020-11-05T17:09:52.0164718 2019-10-01T19:12:47.3489509 Faculty of Science and Engineering School of Engineering and Applied Sciences - Chemistry Fabrizio Pertusati 1 Salvatore Ferla 0000-0002-5918-9237 2 Marcella Bassetto 3 Andrea Brancale 4 Sahar Khandil 5 Andrew D. Westwell 6 Christopher McGuigan 7 |
title |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
spellingShingle |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer Salvatore Ferla Marcella Bassetto |
title_short |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
title_full |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
title_fullStr |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
title_full_unstemmed |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
title_sort |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer |
author_id_str_mv |
d4c62248f510e3b221916989a7bbe6a6 b97beeed16f8e0524551233ade909565 |
author_id_fullname_str_mv |
d4c62248f510e3b221916989a7bbe6a6_***_Salvatore Ferla b97beeed16f8e0524551233ade909565_***_Marcella Bassetto |
author |
Salvatore Ferla Marcella Bassetto |
author2 |
Fabrizio Pertusati Salvatore Ferla Marcella Bassetto Andrea Brancale Sahar Khandil Andrew D. Westwell Christopher McGuigan |
format |
Journal article |
container_title |
European Journal of Medicinal Chemistry |
container_volume |
180 |
container_start_page |
1 |
publishDate |
2019 |
institution |
Swansea University |
issn |
0223-5234 |
doi_str_mv |
10.1016/j.ejmech.2019.07.001 |
publisher |
Elsevier BV |
college_str |
Faculty of Science and Engineering |
hierarchytype |
|
hierarchy_top_id |
facultyofscienceandengineering |
hierarchy_top_title |
Faculty of Science and Engineering |
hierarchy_parent_id |
facultyofscienceandengineering |
hierarchy_parent_title |
Faculty of Science and Engineering |
department_str |
School of Engineering and Applied Sciences - Chemistry{{{_:::_}}}Faculty of Science and Engineering{{{_:::_}}}School of Engineering and Applied Sciences - Chemistry |
url |
http://orca.cf.ac.uk/124785/ |
document_store_str |
0 |
active_str |
0 |
published_date |
2019-10-15T04:04:27Z |
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1763753347407413248 |
score |
11.012678 |