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Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation

Salvatore Ferla Orcid Logo, Mohamed S. Gomaa, Andrea Brancale, Jinge Zhu, Justin T. Ochalek, Hector F. DeLuca, Claire Simons

European Journal of Medicinal Chemistry, Volume: 87, Pages: 39 - 51

Swansea University Author: Salvatore Ferla Orcid Logo

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DOI (Published version): 10.1016/j.ejmech.2014.09.035

Published in: European Journal of Medicinal Chemistry
ISSN: 0223-5234
Published: Elsevier BV 2014
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URI: https://cronfa.swan.ac.uk/Record/cronfa55495
first_indexed 2020-10-23T08:07:51Z
last_indexed 2020-12-11T04:19:47Z
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recordtype SURis
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spelling 2020-12-10T12:08:29.7750369 v2 55495 2020-10-22 Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation d4c62248f510e3b221916989a7bbe6a6 0000-0002-5918-9237 Salvatore Ferla Salvatore Ferla true false 2020-10-22 MEDS Journal Article European Journal of Medicinal Chemistry 87 39 51 Elsevier BV 0223-5234 Imidazole styrylindoles; Sulfonyl styrylindoles; CYP24A1; Vitamin D; Molecular modelling 24 11 2014 2014-11-24 10.1016/j.ejmech.2014.09.035 COLLEGE NANME Medical School COLLEGE CODE MEDS Swansea University 2020-12-10T12:08:29.7750369 2020-10-22T18:32:16.4268896 Faculty of Medicine, Health and Life Sciences Swansea University Medical School - Medicine Salvatore Ferla 0000-0002-5918-9237 1 Mohamed S. Gomaa 2 Andrea Brancale 3 Jinge Zhu 4 Justin T. Ochalek 5 Hector F. DeLuca 6 Claire Simons 7
title Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
spellingShingle Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
Salvatore Ferla
title_short Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_full Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_fullStr Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_full_unstemmed Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_sort Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
author_id_str_mv d4c62248f510e3b221916989a7bbe6a6
author_id_fullname_str_mv d4c62248f510e3b221916989a7bbe6a6_***_Salvatore Ferla
author Salvatore Ferla
author2 Salvatore Ferla
Mohamed S. Gomaa
Andrea Brancale
Jinge Zhu
Justin T. Ochalek
Hector F. DeLuca
Claire Simons
format Journal article
container_title European Journal of Medicinal Chemistry
container_volume 87
container_start_page 39
publishDate 2014
institution Swansea University
issn 0223-5234
doi_str_mv 10.1016/j.ejmech.2014.09.035
publisher Elsevier BV
college_str Faculty of Medicine, Health and Life Sciences
hierarchytype
hierarchy_top_id facultyofmedicinehealthandlifesciences
hierarchy_top_title Faculty of Medicine, Health and Life Sciences
hierarchy_parent_id facultyofmedicinehealthandlifesciences
hierarchy_parent_title Faculty of Medicine, Health and Life Sciences
department_str Swansea University Medical School - Medicine{{{_:::_}}}Faculty of Medicine, Health and Life Sciences{{{_:::_}}}Swansea University Medical School - Medicine
document_store_str 0
active_str 0
published_date 2014-11-24T07:54:19Z
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score 11.047565

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