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A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents
Romeo Romagnoli,
Paola Oliva,
Maria Kimatrai Salvador,
Stefano Manfredini,
Chiara Padroni,
Andrea Brancale,
Salvatore Ferla ,
Ernest Hamel,
Roberto Ronca,
Federica Maccarinelli,
Fatlum Rruga,
Elena Mariotto,
Giampietro Viola,
Roberta Bortolozzi
European Journal of Medicinal Chemistry, Volume: 214, Start page: 113229
Swansea University Author: Salvatore Ferla
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©2021 All rights reserved. All article content, except where otherwise noted, is licensed under a Creative Commons Attribution Non-Commercial No Derivatives License (CC-BY-NC-ND)
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DOI (Published version): 10.1016/j.ejmech.2021.113229
Abstract
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents
Published in: | European Journal of Medicinal Chemistry |
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ISSN: | 0223-5234 |
Published: |
Elsevier BV
2021
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URI: | https://cronfa.swan.ac.uk/Record/cronfa56244 |
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2021-06-24T11:13:07.7231079 v2 56244 2021-02-12 A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents d4c62248f510e3b221916989a7bbe6a6 0000-0002-5918-9237 Salvatore Ferla Salvatore Ferla true false 2021-02-12 PHAR Journal Article European Journal of Medicinal Chemistry 214 113229 Elsevier BV 0223-5234 Antimitotic agents; Structure-activity relationship; 1H-pyrrole; Antiproliferative activity; Tubulin polymerization 15 3 2021 2021-03-15 10.1016/j.ejmech.2021.113229 COLLEGE NANME Pharmacy COLLEGE CODE PHAR Swansea University 2021-06-24T11:13:07.7231079 2021-02-12T11:45:23.4998047 Faculty of Medicine, Health and Life Sciences Swansea University Medical School - Medicine Romeo Romagnoli 1 Paola Oliva 2 Maria Kimatrai Salvador 3 Stefano Manfredini 4 Chiara Padroni 5 Andrea Brancale 6 Salvatore Ferla 0000-0002-5918-9237 7 Ernest Hamel 8 Roberto Ronca 9 Federica Maccarinelli 10 Fatlum Rruga 11 Elena Mariotto 12 Giampietro Viola 13 Roberta Bortolozzi 14 56244__19353__f530d46adb644e9a977cc55dbd95c0d4.pdf 56244.pdf 2021-02-23T16:31:29.5102255 Output 7587066 application/pdf Accepted Manuscript true 2022-01-29T00:00:00.0000000 ©2021 All rights reserved. All article content, except where otherwise noted, is licensed under a Creative Commons Attribution Non-Commercial No Derivatives License (CC-BY-NC-ND) true eng https://creativecommons.org/licenses/by-nc-nd/4.0/ |
title |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
spellingShingle |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents Salvatore Ferla |
title_short |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
title_full |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
title_fullStr |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
title_full_unstemmed |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
title_sort |
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents |
author_id_str_mv |
d4c62248f510e3b221916989a7bbe6a6 |
author_id_fullname_str_mv |
d4c62248f510e3b221916989a7bbe6a6_***_Salvatore Ferla |
author |
Salvatore Ferla |
author2 |
Romeo Romagnoli Paola Oliva Maria Kimatrai Salvador Stefano Manfredini Chiara Padroni Andrea Brancale Salvatore Ferla Ernest Hamel Roberto Ronca Federica Maccarinelli Fatlum Rruga Elena Mariotto Giampietro Viola Roberta Bortolozzi |
format |
Journal article |
container_title |
European Journal of Medicinal Chemistry |
container_volume |
214 |
container_start_page |
113229 |
publishDate |
2021 |
institution |
Swansea University |
issn |
0223-5234 |
doi_str_mv |
10.1016/j.ejmech.2021.113229 |
publisher |
Elsevier BV |
college_str |
Faculty of Medicine, Health and Life Sciences |
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facultyofmedicinehealthandlifesciences |
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Faculty of Medicine, Health and Life Sciences |
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facultyofmedicinehealthandlifesciences |
hierarchy_parent_title |
Faculty of Medicine, Health and Life Sciences |
department_str |
Swansea University Medical School - Medicine{{{_:::_}}}Faculty of Medicine, Health and Life Sciences{{{_:::_}}}Swansea University Medical School - Medicine |
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published_date |
2021-03-15T04:11:03Z |
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11.028886 |